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CAS:43229-80-7|Formoterol Hemifumarate

发布时间:2022-03-17     作者:德尔塔   分享到:

【产品介绍】:

产品名称 Formoterol Hemifumarate 英文名称 Formoterol Hemifumarate 应用 A potent β2-AR agonist. 规格或纯度 ≥99% 别名 富马酸福莫特罗 英文别名 Foradil;N-[2-Hydroxy-5-[[(1RS)-1-hydroxy-2-[[(1RS)-2-(4-methoxyphenyl)-1-methylethyl]amino]ethyl]phenyl]formamide (E)-2-butenedioate 运输条件 冰袋运输 生化机理 Formoterol Fumarate is shown to be a potent β-AR adrenoceptor agonist, with a fast onset of effect on the isolated human bronchus model. This compound demonstrates a 330-fold selectivity for β2 over β1 receptors. Formoterol Fumarate has been reported to be 150-200 times more potent than isoprenaline. This agent has also been noted to reduce the loss of muscle mass in murine models.Potent long-acting β 2 adrenoceptor agonist. K i values are 27 and 2400 nM for adrenergic receptor subtypes β 2 and β 1 , respectively. Trachea muscle relaxant.CAS编号 43229-80-7 溶解性 DMSO 80 mg/mL Water Ethanol 储存温度 2-8°C储存 分子量 402.4 分子式 C19H24N2O4·1/2C4H4O4 PubChem CID 53477580