「同位素标记抑制剂」CAS:1246817-44-6|Dabigatran-d3
【产品介绍】:
生物活性:Dabigatran-d3 is the deuterium labeled Dabigatran. Dabigatran (BIBR 953), an oral anticoagulant, is a reversible, potent, competitive direct thrombin inhibitor (Ki=4.5 nM). Dabigatran (BIBR 953) also inhibits thrombin-induced platelet aggregation (IC50=10 nM)[1][2].
体外研究(In Vitro):Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].
德尔塔生物 has not independently confirmed the accuracy of these methods. They are for reference only.
Dabigatran-d3 相关抗体:
PAR2 Antibody (YA2455)
Protein C Antibody (YA2461)
Thrombomodulin Antibody (YA891)
Thrombomodulin Antibody (YA892)
F2 Antibody
PAR6 Antibody (YA1536)
Prothrombin Antibody (YA1753)
PAR4 Antibody (YA2603)
Protein S Antibody (YA2919)
分子量:474.53
Formula:C25H22D3N7O3
CAS 号:1246817-44-6
非标记 CAS:211914-51-1
性状:固体
颜色:Off-white to light yellow
中文名称:达比加群 d3
运输条件:Room temperature in continental US; may vary elsewhere.
储存方式:Powder:-20°C:3 years,4°C:2 years
In solvent:-80°C:6 months,-20°C:1 month