德尔塔
您当前所在位置:首页 > 宣传资料 > 材料科学 > 荧光材料

「同位素标记抑制剂」CAS:2140316-62-5|Vortioxetine-d8

发布时间:2025-06-13     作者:德尔塔生物   分享到:

【产品介绍】:

生物活性:Vortioxetine-d8 (Lu AA 21004-d8) is a deuterated version of Vortioxetine. Vortioxetine (Lu AA 21004) is an antagonist of 5-HT3A and 5-HT7 receptors (Ki: 3.7 nM, 19 nM) and an inhibitor of 5-hydroxytryptamine transporter (SERT) (Ki: 1.6 nM), as well as a 5-HT1A agonist and a partial 5-HT1B agonist (Ki: 15 nM, 33 nM)[1].
分子量:306.49
Formula:C18H14D8N2S
CAS 号:2140316-62-5
非标记 CAS:508233-74-7
中文名称:沃替西汀 d8
运输条件:Room temperature in continental US; may vary elsewhere.
储存方式:Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
Data Sheet (528 KB)
产品使用指南 (1538 KB)
参考文献
[1]. Bang-Andersen B, et al. Discovery of 1-[2-(2,4-dimethylphenylsulfanyl)phenyl]piperazine (Lu AA21004): a novel multimodal compound for the treatment of major depressive disorder. J Med Chem. 2011 May 12;54(9):3206-21.
 [Content Brief]