德尔塔
您当前所在位置:首页 > 分析科学 > 全部产品

「同位素标记抑制剂」(S)-Mirtazapine-d3

发布时间:2025-09-23     作者:德尔塔生物   分享到:

【产品介绍】:

生物活性:(S)-Mirtazapine-d3 is a deuterium labeled (S)-Mirtazapine. (S)-Mirtazapine is a S(+)-enantiomer of Mirtazapine with pronociceptive properties in an animal model of acute thermal nociception.(S)-Mirtazapine is a stereoselective 5-HT2 receptor antagonist. (S)-Mirtazapine is metabolized by CYP2D6 and CYP1A2[1].
IC50 & Target:5-HT2 receptor[1]
分子量:268.37
Formula:C17H16D3N3
非标记 CAS:61337-87-9
性状:固体
颜色:White to off-white
中文名称:米氮平杂质13 d4-d3
运输条件:Room temperature in continental US; may vary elsewhere.
储存方式:Powder:-20°C:3 years,4°C:2 years
In solvent:-80°C:6 months,-20°C:1 month
纯度 & 产品资料
纯度: ≥99.0%
参考文献
[1]. Muth-Selbach U, et al. Racemic intrathecal mirtazapine but not its enantiomers acts anti-neuropathic after chronic constriction injury in rats. Brain Res Bull. 2009 Apr 6;79(1):63-8.
 [Content Brief]