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CAS:786686-79-1|Olanzapine-d3,奥氮平 D3; LY170053-d3

发布时间:2025-06-10     作者:德尔塔生物   分享到:

【产品介绍】:

生物活性:Olanzapine-d3 is the deuterium labeled Olanzapine. Olanzapine is a selective, orally active monoaminergic antagonist with high affinity binding to serotonin H1, 5HT2A/2C, 5HT3, 5HT6 (Ki=7, 4, 11, 57, and 5 nM, respectively), dopamine D1-4 (Ki=11 to 31 nM), muscarinic M1-5 (Ki=1.9-25 nM), and adrenergic α1 receptors (Ki=19 nM). Olanzapine is an atypical antipsychotic[1][2].
IC50 & Target:D3 Receptor
mAChR1
分子量:315.45
Formula:C17H17D3N4S
CAS 号:786686-79-1
非标记 CAS:132539-06-1
性状:固体
颜色:White to yellow
中文名称:奥氮平 d3;奥兰氮平 d3
运输条件:Room temperature in continental US; may vary elsewhere.
储存方式:Powder:-20°C:3 years,4°C:2 years
In solvent:-80°C:6 months,-20°C:1 month